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DEVANIB

DEUCRAVACITINIB · by HORIZON

ANTINEOPLASTICS Tyrosine kinase 2 (TYK2) inhibitor HORIZON

Composition

Tab: Deucravacitinib 6 mg

Indications & Dosage

Treatment of moderate to severe plaque psoriasis in adult candidate for systemic therapy or phototherapy: Adult: 6 mg once daily, dose should be taken at the same time every day with or without meal.

Contraindications

Severe hepatic impairment (Child-Pugh C), hypersensitivity reaction (angioedema).

Precautions

Increased risk of infection, evaluate patients for tuberculosis prior to initiating treatment if positive consider treating tuberculosis before starting Deucravacitinib. Periodically evaluate serum triglyceride level and liver enzymes levels.

Interactions

Aliskiren, Antacids, Antiarrhythmics, Antiepileptics, Antifungals, azoles, non-sedating antihistamines, Aprepitant, Calcium channel blockers, ciclosporin, Cobicistat, colchicine, Coumarins (warfarin), Crizotinib, dabigatran, digoxin, edoxaban, Enzalutamide, ergotamine, everolimus, Grapefruit juice (avoid), H2 receptor antagonists, HIV-protease inhibitors, Idelalisib, Imatinib, Lapatinib, loperamide, Macrolides, Netupitant, Nilotinib, NSAIDs, Opioids, pimozide, Proton pump inhibitors, Ranolazine, Rifampicin, sirolimus. St Johns Wort, sulfonylureas (glimepiride). Tacrolimus, Taxanes, topotecan.

Pregnancy

Avoid unless essential

Lactation

Contraindicated. Discontinue breast-feeding

Side Effects

Increased risk of infection, Malignancy including lymphoma, upper respiratory infection, herpes simplex, mouth ulcer, increased triglyceride level, increased liver enzymes