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ERTULIX-S

ERTUGLIFLOZIN AND SITAGLIPTIN · by HELIX

BLOOD GLUCOSE LOWERING DRUGS, EXCLUDING INSULIN Sodium Glucose Co-transporter 2 (SGLT2) Inhibitors/Dipeptidylpeptidase-4 Inhibitors HELIX

Composition

Tab 5/100 mg/15/100 mg: Ertugliflozin 5 mg/15 mg and 100 mg Sitagliptin

Indications & Dosage

Type 2 diabetes mellitus if monotherapy fails to achieve adequate glycaemic control: Adult: 5/100 mg once daily; increased to 15/100 mg once daily if required, dose to be taken in the morning.

Contraindications

Severe renal impairment, end-stage renal disease, or dialysis, Pancreatitis, Ketoacidosis

Precautions

Heart failure, renal impairment, hypotension, urosepsis and pyelonephritis, genital mycotic infection, increase LDL-C, severe arthralgia, pemphigoid, peripheral vascular disease, neuropathy, diabetic foot ulcer, high cholesterol level, gallstones.

Pregnancy

Contraindicated in pregnancy

Lactation

Contraindicated or not recommended

Side Effects

Hypoglycaemia, hypovolaemia, increased risk of infection, polydipsia, thirst, urinary disorders, vulvovaginal pruritus. Rare: Diabetic ketoacidosis (discontinue), Fourniers gangrene (discontinue). lower limb amputations, phimosis