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LAMRIN

LAMIVUDINE · by PHARMEDIC

ANTIVIRALS FOR SYSTEMIC USE Nucleoside reverse transcriptase inhibitor PHARMEDIC

Composition

Tab 100 mg/150 mg: Lamivudine 100 mg/150 mg. Oral Soln 5 mg/10 mg: Per ml: Lamivudine 5 mg/10 mg.

Indications & Dosage

HIV infection in combination with other antiretroviral drugs: Adult: 150 mg every 12 hours, alternatively 300 mg once daily preferably without food. Children above 3 months: 4 mg/ kg twice daily, max 300 mg daily.

Precautions

Renal impairment; reduce dose, advanced liver disease due to Hepatitis B, pancreatitis.Recurrent hepatitis in patients with chronichepatitis B may occur on discontinuation of lamivudine.Initiate treatment under specialist supervision.

Interactions

IV ganciclovir, foscarnet, co-trimoxazole.

Pregnancy

Caution advised

Lactation

Caution advised, avoid

Side Effects

Alopecia, muscle disorders, nasal symptoms, peripheral neuropathy, rhabdomyolysis, neutropenia, anaemia, thrombocytopenia, raised liver enzymes, serum amylase, headache, malaise, fatigue, GI disturbance, abdominal pain, insomnia, cough, musculoskeletal pain, pancreatitis,