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Composition

Tab 10 mg/20 mg: Zafirlukast 10 mg/20 mg.

Indications & Dosage

Prophylaxis and treatment of asthma: Adult & Children above 12 yrs: 20 mg twice daily.

Contraindications

Hepatic impairment, cirrhosis, hypersensitivity.

Precautions

Moderate to severe renal impairment, elderly, risk of eosinophilic condition or a Churg-Strauss syndrome; discontinue if occur. If signs or symptoms of hepatotoxicity; measure serum transaminases and consider withdrawing therapy.

Interactions

Warfarin, theophylline, aspirin, terfenadine, erythromycin, smoking.

Pregnancy

Not known to be harmful

Lactation

Caution advised

Side Effects

Abdominal pain, GI disturbances, headache, respiratory infections, insomnia, malaise, hypersensitivity reactions Rare: Angioedema, arthralgia, bleeding disorders, hepatitis, hyperbilirubinaemia, myalgia, skin reactions, thrombocytopenia, agranulocytosis, Churg-Strauss syndrome (Discontinue)