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NEXAVAR

SORAFENIB · by BAYER

ANTINEOPLASTICS Protein kinase inhibitor BAYER

Composition

Tab 200 mg: Sorafenib 200 mg.

Indications & Dosage

Treatment of advanced renal cell carcinoma when treatment with interferon alfa or interleukin-2 has failed or is unsuitable, Treatment of progressive, locally advanced, or metastatic, differentiated thyroidcarcinoma that is refractory to radioactive iodine, Treatment of hepatocellular carcinoma: Adult: 400 mg twice daily, for dose adjustments due toside effects, consult product literature. Children: Not recommended.

Precautions

Cardiac ischaemia, major surgical procedures, potential risk of bleeding; treat tracheal, bronchial, oroesophageal infiltration with localized therapy before initiating treatment, consider permanent withdrawal if patient requires medical intervention for bleeding, susceptibility to QT-interval prolongation, dermatological toxicities, hemorrhage, infarction, wound healing complications, GI perforation, hepatic impairment.

Interactions

Warfarin, irinotecan, docetaxel, rifampicin, phe-nytoin, carbamazepine, phenobarb, dexamethasone, St. Johns wort, doxorubicin.

Pregnancy

Contraindicated in pregnancy.

Lactation

Contraindicated. Discontinue breast-feeding

Side Effects

Anorexia, arthralgia, asthenia, congestive heart failure, depression, dermatitis, desquamation, dysgeusia, dyspepsia, dysphagia, dysphonia, erythema, fatigue, flushing, GI upset, gastro-oesophageal reflux disease, haemorrhage, hand-foot skin reaction, hyperkeratosis, hypertension, hypophosphataemia, hypophosphataemia, keratoacanthoma, malaise, muscle spasms, myalgia, myocardial infarction, myocardialischaemia, peripheral neuropathy, proteinuria, pruritus, rash, renal failure, rhinorrhea, thyroid dysfunction, tinnitus, alopecia, bone-marrow suppression, hyperuricaemia, nausea, oral mucositis, thromboembolism, tumourlysis syndrome, vomiting